Felypressin acetate

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Felypressinacetate 是 vasopressin 1 的激动剂，作用于所有精氨酸 vasopressin 受体 1AS。醋酸铁加压素可用于牙科手术。

Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.(In Vitro):Felypressin is a synthetic hormone of the posterior pituitary lobe characterized by vasoconstrictor properties mediated by V1 receptors of the blood vessel smooth muscle cells.(In Vivo):In Wistar rats, Felypressin (240 ng/kg; i.v.) induces a pressor effect and bradycardic effect depending on V1 receptors to induce pressor and bradycardic effects. Felypressin produces a high relationship between bradycardia and mean arterial pressure variation depending on area postrema and central V1 receptors. Felypressin reduces toxicity during dental procedures. Felypressin increases the diastolic blood pressure of hypertensive patients with controlled blood pressure.

Felypressin is a synthetic hormone of the posterior pituitary lobe characterized by vasoconstrictor properties that is widely used in dental procedures. The vasoconstrictor action of Felypressin seems to be mediated by V1 receptors of the blood vessel smooth muscle cells.

Felypressin can reduce toxicity during dental procedures. Felypressin increases the diastolic blood pressure of hypertensive patients with controlled blood pressure. Cardiovascular effects of Felypressin (240 ng/kg; intravenous injection) are studied in Wistar rats. Felypressin induces a pressor effect. Felypressin depends on V1 receptors to induce pressor and bradycardic effects, and that it produces a high relationship between bradycardia and mean arterial pressure variation depending on area postrema and central V1 receptors.

PLV-2 acetate

GPCR/G Protein

Vasopressin Receptor

MEK1|MEK2|Autophagy|Mitophagy

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914453-97-7

1100.28

C48H69N13O13S2

>98% (HPLC)

In Vitro:?H2O : 100 mg/mL

CC(O)=O.NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O

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(-20℃)

With Ice Pack

≥ 2 years